Gene
|
CPT Code(s)
|
Generic Name
|
Trade Name(s)
|
Intended use for Drug(s)
|
Guidance
|
BCHE
|
81479
|
mivacurium, succinylcholine
|
Mivacurium chloride, Anectine
|
Neuromuscular blocking agent
|
FDA
|
CACNA1S
|
81479
|
desflurane, enflurane, halothane, isoflurane, methoxyflurane, sevoflurane, succinylcholine
|
Suprane, Ethrane, Fluothane, Forane, Penthrox, Ultane, Anectine, Quelicin
|
Volatile anesthetic
|
CPIC
|
CFTR
|
81220
|
ivacaftor
|
Kalydeco
|
Cystic fibrosis
|
CPIC
|
CYP2B6
|
81479
|
efavirenz
|
Sustiva
|
Antiretroviral; HIV
|
CPIC/FDA
|
CYP2C19
|
81225
|
brivaracetam, clobazam
|
Briviact, Onfi
|
Anticonvulsant
|
FDA
|
CYP2C19
|
81225
|
citalopram, escitalopram, sertraline
|
Celexa, Lexapro, Zoloft
|
Antidepressant - Selective Serotonin Reuptake Inhibitor (SSRI)
|
CPIC/FDA
|
CYP2C19
|
81225
|
amitriptyline, clomipramine, doxepin, imipramine, trimipramine
|
Elavil, Anafranil, Silenor, Tofranil, Surmontil
|
Antidepressant - Tricyclic
|
CPIC
|
CYP2C19
|
81225
|
voriconazole
|
Vfend
|
Antifungal
|
CPIC/FDA
|
CYP2C19
|
81225
|
flibanserin
|
Addyi
|
Mixed serotonin agonist
|
FDA
|
CYP2C19
|
81225
|
clopidogrel
|
Plavix
|
Platelet aggregation inhibitor
|
CPIC/FDA
|
CYP2C19
|
81225
|
dexlansoprazole, lansoprazole, omeprazole, pantoprazole
|
Dexilant, Prevacid, Prilosec, Protonix
|
Proton Pump Inhibitor (PPI)
|
CPIC/FDA
|
CYP2C9
|
81227
|
warfarin
|
Jantoven, Coumadin
|
Anticoagulant
|
CPIC/FDA
|
CYP2C9
|
81227
|
fosphenytoin, phenytoin
|
Cerebyx, Dilantin
|
Anticonvulsant
|
CPIC/FDA
|
CYP2C9
|
81227
|
dronabinol
|
Marinol, Syndros
|
Antiemetic
|
FDA
|
CYP2C9
|
81227
|
erdafitinib
|
Balversa
|
FGFR kinase inhibitor, bladder cancer
|
FDA
|
CYP2C9
|
81227
|
siponimod
|
Mayzent
|
Multiple sclerosis
|
FDA
|
CYP2C9
|
81227
|
celecoxib, flurbiprofen, lornoxicam, meloxicam, piroxicam, tenoxicam
|
Celebrex, Ansaid, Ocufen, Chlortenoxicam, Xefo, Mobic, Vivlodex, Anjeso, Qmiiz ODT, Feldene, Mobiflex
|
Non-steroidal anti-inflammatory (NSAID)
|
CPIC/FDA
|
CYP2D6
|
81226, 0070U,
0071U, 0072U,
0073U, 0074U, 0075U, 0076U
|
carvedilol
|
Coreg
|
Alpha - Beta blocker
|
FDA
|
CYP2D6
|
81226, 0070U,
0071U, 0072U,
0073U, 0074U,
0075U, 0076U
|
propafenone
|
Rythmol
|
Antiarrhythmic
|
FDA
|
CYP2D6
|
81226, 0070U,
0071U, 0072U,
0073U, 0074U,
0075U, 0076U
|
fluvoxamine, paroxetine, venlafaxine, vortioxetine
|
Luvox, Paxil, Effexor XR, Brintellix, Trintellix
|
Antidepressant – Selective Serotonin Reuptake Inhibitor (SSRI)
|
CPIC/FDA
|
CYP2D6
|
81226, 0070U,
0071U, 0072U,
0073U, 0074U,
0075U, 0076U
|
amitriptyline, clomipramine, desipramine, doxepin, imipramine, nortriptyline, trimipramine
|
Elavil, Anafranil, Norpramin, Silenor, Tofranil, Aventyl, Pamelor, Surmontil
|
Antidepressant - Tricyclic
|
CPIC
|
CYP2D6
|
81226, 0070U,
0071U, 0072U,
0073U, 0074U,
0075U, 0076U
|
meclizine, ondansetron, tropisetron
|
Antivert, Zofran ODT, Tropisetron
|
Antiemetic
|
CPIC/FDA
|
CYP2D6
|
81226, 0070U,
0071U, 0072U,
0073U, 0074U,
0075U, 0076U
|
gefitinib, tamoxifen
|
Iressa, Soltamox, Nolvadex
|
Antineoplastic
|
CPIC/FDA
|
CYP2D6
|
81226, 0070U,
0071U, 0072U,
0073U, 0074U,
0075U, 0076U
|
aripiprazole, aripiprazole lauroxil, brexpiprazole, clozapine, iloperidone, perphenazine, pimozide, thioridazine
|
Abilify, Aristada, Rexulti, Clozaril, FazaClo, Versacloz, Fanapt, Trilafon, Orap, Mellaril
|
Antipsychotic
|
FDA
|
CYP2D6
|
81226, 0070U,
0071U, 0072U,
0073U, 0074U,
0075U, 0076U
|
amphetamine, atomoxetine
|
Adzenys ER, Dyanavel XR, Adderall, Strattera
|
Attention Deficit - Hyperactivity (ADHD) Therapy
|
CPIC/FDA
|
CYP2D6
|
81226, 0070U,
0071U, 0072U,
0073U, 0074U,
0075U, 0076U
|
metoclopramide
|
Reglan
|
Gastrointestinal prokinetic agent
|
FDA
|
CYP2D6
|
81226, 0070U,
0071U, 0072U,
0073U, 0074U,
0075U, 0076U
|
eliglustat
|
Cerdelga
|
Gaucher's disease
|
FDA
|
CYP2D6
|
81226, 0070U,
0071U, 0072U,
0073U, 0074U,
0075U, 0076U
|
deutetrabenazine, tetrabenazine
|
Austedo, Xenazine
|
Movement disorder therapy
|
FDA
|
CYP2D6
|
81226, 0070U,
0071U, 0072U,
0073U, 0074U,
0075U, 0076U
|
pitolisant
|
Wakix
|
Narcolepsy therapy agent
|
FDA
|
CYP2D6
|
81226, 0070U,
0071U, 0072U,
0073U, 0074U,
0075U, 0076U
|
codeine, oliceridine, tramadol
|
Olinvyk, Ultram
|
Opioid
|
CPIC/FDA
|
CYP2D6
|
81226, 0070U,
0071U, 0072U,
0073U, 0074U,
0075U, 0076U
|
lofexidine
|
Lucemyra
|
Opioid withdrawal
|
FDA
|
CYP2D6
|
81226, 0070U,
0071U, 0072U,
0073U, 0074U,
0075U, 0076U
|
cevimeline
|
Evoxac
|
Saliva stimulant
|
FDA
|
CYP2D6
|
81226, 0070U,
0071U, 0072U,
0073U, 0074U,
0075U, 0076U
|
tolterodine
|
Detrol
|
Urinary antispasmodic
|
FDA
|
CYP2D6
|
81226, 0070U,
0071U, 0072U,
0073U, 0074U,
0075U, 0076U
|
valbenazine
|
Ingrezza
|
VMAT2 inhibitor
|
FDA
|
CYP3A5
|
81231
|
tacrolimus
|
Prograf
|
Antirejection
|
CPIC/FDA
|
CYP4F2
|
81479
|
warfarin
|
Jantoven, Coumadin
|
Anticoagulant
|
CPIC/FDA
|
DPYD
|
81232
|
capecitabine, fluorouracil
|
Xeloda, Adrucil, Efudex, Fluoroplex, Tolak
|
Antineoplastic
|
CPIC/FDA
|
G6PD
|
81247
|
rasburicase
|
Elitek
|
Hyperuricemia
|
CPIC
|
HLA - A
|
81381, 81374
|
carbamazepine
|
Tegretol
|
Anticonvulsant
|
CPIC/FDA
|
HLA-A
|
81381
|
tebentafusp
|
Kimmtrak
|
antineoplastic
|
FDA
|
HLA - B
|
81381, 81374
|
carbamazepine, fosphenytoin, oxcarbazepine, phenytoin
|
Tegretol, Cerebyx, Trileptal, Dilantin
|
Anticonvulsant
|
CPIC/FDA
|
HLA - B
|
81381, 81374
|
pazopanib
|
Votrient
|
Antineoplastic
|
FDA
|
HLA - B
|
81381, 81374
|
abacavir
|
Ziagen
|
Antiretroviral; HIV
|
CPIC/FDA
|
HLA - B
|
81381, 81374
|
allopurinol
|
Aloprim, Zyloprim
|
Hyperuricemia
|
CPIC/FDA
|
HLA - DQA1
|
81377, 81383
|
lapatinib
|
Tykerb
|
Antineoplastic
|
FDA
|
HLA - DRB1
|
81377, 81383
|
lapatinib
|
Tykerb
|
Antineoplastic
|
FDA
|
IFNL3
|
81283
|
peginterferon alfa - 2a, peginterferon alfa - 2b
|
Pegasys, Pegasys ProClick, PegIntron, Sylatron
|
Antiviral, HCV
|
CPIC
|
NAT2
|
81479
|
procainamide
|
Procan, Pronestyl
|
Antiarrhythmic
|
FDA
|
NAT2
|
81479
|
sulfamethoxazole / trimethoprim
|
Bactrim
|
Antibacterial
|
FDA
|
NAT2
|
81479
|
isoniazid
|
Niazid
|
Antitubercular
|
FDA
|
NAT2
|
81479
|
sulfasalazine
|
Azulfidine
|
Disease-Modifying Antirheumatic Drug (DMARD): Other - inflammatory bowel agent
|
FDA
|
NAT2
|
81479
|
amifampridine, amifampridine phosphate
|
Ruzurgi, Firdapse
|
Multiple sclerosis
|
FDA
|
NUDT15
|
81306
|
azathioprine, mercaptopurine, thioguanine
|
Azasan, Purixan, Tabloid
|
Antineoplastic
|
CPIC/FDA
|
RYR1
|
81406
|
desflurane, enflurane, halothane, isoflurane, methoxyflurane, sevoflurane, succinylcholine
|
Suprane, Ethrane, Fluothane, Forane, Penthrox, Ultane, Anectine, Quelicin
|
Volatile anesthetic
|
CPIC
|
SLCO1B1
|
81328
|
simvastatin
|
FloLipid, Zocor
|
Antihyperlipidemic
|
CPIC/FDA
|
TPMT
|
81335, 0034U, 0286U
|
azathioprine, mercaptopurine, thioguanine
|
Azasan, Purixan, Tabloid
|
Antineoplastic
|
CPIC/FDA
|
UGT1A1
|
81350
|
belinostat, irinotecan, nilotinib, pazopanib, Sacituzumab Govitecan - hziy
|
Beleodaq, Camptosar, Tasigna, Votrient, Trodelvy
|
Antineoplastic
|
FDA
|
UGT1A1
|
81350
|
atazanavir
|
Reyataz
|
Antiretroviral, HIV
|
CPIC
|
VKORC1
|
81355
|
warfarin
|
Jantoven, Coumadin
|
Anticoagulant
|
CPIC/FDA
|